Translation for "reseptori" to english
Translation examples
Farmakologisella tasolla, atsapironit sitoutuvat seuraaviin reseptoreihin eri suhteissa: 5-HT1A-reseptori (osittais- tai täyagonisti) 5-HT2A-reseptori (käänteisagonisti) D2-reseptori (antagonisti tai osittaisagonisti) α1-reseptori (antagonisti) α2-reseptori (antagonisti) Jotkin atsapironit sitoutuvat myös D4, 5-HT2C, 5-HT7, and sigmareseptoreihin.
On a pharmacological level, azapirones varyingly possess activity at the following receptors: 5-HT1A receptor (as partial or full agonists) 5-HT2A receptor (as inverse agonists) D2 receptor (as antagonists or partial agonists) α1-adrenergic receptor (as antagonists) α2-adrenergic receptor (as antagonists) Actions at D4, 5-HT2C, 5-HT7, and sigma receptors have also been shown for some azapirones.
Se sitoutuu CB1-reseptoriin noin viisi kertaa voimakkaammin kuin CB2-reseptoriin.
It binds primarily to the CB1 receptor, and only weakly to the CB2 receptor.
Palautumaton antagonisti sitoutuu kovalenttisesti reseptoriin estäen muiden ligandien reseptoriin sitoutumisen.
An irreversible antagonist binds so strongly to the receptor as to render the receptor unavailable for binding to the agonist.
Losartaanin vaikutus perustuu angiotensiini II -reseptorien eli AT-reseptorien toiminnan estämiseen.
The action of AII itself is targeted by angiotensin II receptor antagonists, which directly block angiotensin II AT1 receptors.
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